adrenergic receptor chart

Receptor type

Agonist potency orderSelected action

of agonistAgonists Antagonists

α1adrenaline ≥ noradrenaline >> isoprenaline

smooth muscle contraction

(Alpha-1 agonists)

Noradrenaline Phenylephrine Methoxamine Cirazoline

Xylometazoline

(Alpha-1 blockers) Doxazosin Phenoxybenzamine Phentolamine Prazosin Tamsulosin

Terazosin

α2adrenaline ≥ noradrenaline >> isoprenaline

smooth muscle contraction and neurotransmitter inhibition

(Alpha-2 agonists)

Clonidine Guanafacin Monoxidine Alpha.methydopa

Guanfacine

(Alpha-2 blockers) Yohimbine Idazoxan Tolazoline Rauwolscine

.

β1isoprenaline > adrenaline = noradrenaline

heart muscle contraction

Noradrenaline Isoprenaline

Dobutamine

Metoprolol

Atenolol

β2isoprenaline > adrenaline >> noradrenaline

smooth muscle relaxation

Salbutamol , Albuterol Bitolterol mesylate Formoterol Isoprenaline Levalbuterol Metaproterenol Salmeterol Terbutaline

Ritodrine

(Beta blockers) Butoxamine Propranolol Nadolol Carteolol Timolol Sotalol

β3isoprenaline = noradrenaline > adrenaline

Enhance lipolysis Amibegron

Solabegron

http://en.wikipedia.org/wiki/Solabegron

http://en.wikipedia.org/wiki/Amibegron

http://en.wikipedia.org/wiki/Lipolysis

http://en.wikipedia.org/wiki/Beta-3_adrenergic_receptor

http://en.wikipedia.org/wiki/Propranolol

http://en.wikipedia.org/wiki/Butoxamine

http://en.wikipedia.org/wiki/Beta_blocker

http://en.wikipedia.org/wiki/Ritodrine

http://en.wikipedia.org/wiki/Terbutaline

http://en.wikipedia.org/wiki/Salmeterol

http://en.wikipedia.org/wiki/Metaproterenol

http://en.wikipedia.org/wiki/Levalbuterol

http://en.wikipedia.org/wiki/Isoprenaline

http://en.wikipedia.org/wiki/Formoterol

http://en.wikipedia.org/wiki/Bitolterol_mesylate

http://en.wikipedia.org/wiki/Albuterol

http://en.wikipedia.org/wiki/Salbutamol


http://en.wikipedia.org/wiki/Atenolol

http://en.wikipedia.org/wiki/Metoprolol

http://en.wikipedia.org/wiki/Dobutamine


http://en.wikipedia.org/wiki/Noradrenaline

http://en.wikipedia.org/wiki/Heart_muscle


http://en.wikipedia.org/wiki/Idazoxan

http://en.wikipedia.org/wiki/Yohimbine

http://en.wikipedia.org/wiki/Alpha-2_blocker

http://en.wikipedia.org/wiki/Guanfacine

http://en.wikipedia.org/wiki/Lofexidine

http://en.wikipedia.org/wiki/Clonidine

http://en.wikipedia.org/wiki/Alpha-adrenergic_agonist#.CE.B12_agonists

http://en.wikipedia.org/wiki/Smooth_muscle

http://en.wikipedia.org/wiki/Alpha-2_adrenergic_receptor

http://en.wikipedia.org/wiki/Terazosin

http://en.wikipedia.org/wiki/Tamsulosin

http://en.wikipedia.org/wiki/Prazosin

http://en.wikipedia.org/wiki/Phentolamine

http://en.wikipedia.org/wiki/Phenoxybenzamine

http://en.wikipedia.org/wiki/Doxazosin

http://en.wikipedia.org/wiki/Alpha-1_blocker

http://en.wikipedia.org/wiki/Xylometazoline

http://en.wikipedia.org/wiki/Cirazoline

http://en.wikipedia.org/wiki/Methoxamine

http://en.wikipedia.org/wiki/Phenylephrine

http://en.wikipedia.org/wiki/Noradrenaline

http://en.wikipedia.org/wiki/Alpha-adrenergic_agonist#.CE.B11_agonists

http://en.wikipedia.org/wiki/Smooth_muscle


http://en.wikipedia.org/wiki/Alpha-1_adrenergic_receptor

http://en.wikipedia.org/wiki/Adrenergic_antagonist

http://en.wikipedia.org/wiki/Adrenergic_agonist

http://en.wikipedia.org/wiki/Agonist

adrenergic receptor chart

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