contents volume 76 (2001)

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Journal of Controlled Release 76 (2001) 385–387 www.elsevier.com / locate / jconrel Contents Volume 76 (2001) Vol. 76, Nos.1 2 (11 SEPTEMBER 2001) Research papers Effect of PSC 833 liposomes and Intralipid on the transport of epirubicin in Caco-2 cells and rat intestines 1 Yu.-l. Lo, F.-i. Liu, J.-y. Cherng ( Tainan, Taiwan) Protein delivery from materials formed by self-selective conjugate addition reactions 11 D.L. Elbert, A.B. Pratt, M.P . Lutolf , S. Halstenberg, J. A. Hubbell ( Zurich, Switzerland) Temperature-controlled content release from liposomes encapsulating Pluronic F127 27 P . Chandaroy, A. Sen, S. W . Hui ( Buffalo, NY, USA) Investigation of the influence of mean HPMC particle size and number of polymer particles on the release of aspirin from swellable hydrophilic matrix tablets P . W .S. Heng, L. W . Chan, M.G. Easterbrook, X. Li ( Kent Ridge Crescent, Merchant Square, Singapore) 39 Cross-linked high amylose starch derivatives as matrices for controlled release of high drug loadings ´ J. Mulhbacher, P . Ispas-Szabo, V . Lenaerts, M. A. Mateescu ( Montreal, Laval, Canada) 51 Evaluation of particle uptake in human blood monocyte-derived cells in vitro. Does phagocytosis activity of dendritic cells measure up with macrophages? L. Thiele, B. Rothen-Rutishauser, S. Jilek, H. Wunderli- Allenspach, H.P . Merkle, E. Walter ( Zurich, Switzerland) 59 Piroxicam delivery into human stratum corneum in vivo: iontophoresis versus passive diffusion ` C. Curdy, Y.N. Kalia, A. Naik, R.H. Guy (Archamps, France, Geneve, Switzerland) 73 Toxicological evaluation of a bioadhesive nasal powder containing a starch and Carbopol 974 P on rabbit nasal mucosa and slug mucosa C. Callens, E. Adriaens, K. Dierckens, J.P . Remon ( Gent, Belgium) 81 Experimental determination of the theophylline diffusion coefficient in swollen sodium-alginate membranes M. Grassi, I. Colombo, R. Lapasin ( Trieste, Milan, Italy) 93 Poly(ethylene glycol)–human serum albumin–paclitaxel conjugates: preparation, characterization and pharmacokinetics F. Dosio, S. Arpicco, P . Brusa, B. Stella, L. Cattel ( Turin, Italy) 107 Emulsions containing partially water-miscible solvents for the preparation of drug nanosuspensions M. Trotta, M. Gallarate, F. Pattarino, S. Morel ( Novara, Italy) 119 Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in the human intestinal Caco-2 cell line C. U. Nielsen, R. Andersen, B. Brodin, S. Frokjaer, M.E. Taub, B. Steffansen ( Copenhagen, Denmark) 129 Functional feature of a novel model of blood brain barrier: studies on permeation of test compounds A. Cestelli, C. Catania, S. DAgostino, I. Di Liegro, L. Licata, G. Schiera, G.L. Pitarresi, G. Savettieri, V . De Caro, G. Giandalia, L.I. Giannola ( Palermo, Italy) 139 Gene delivery Hydrophilic poly(DL-lactide-co-glycolide) microspheres for the delivery of DNA to human-derived macrophages and dendritic cells E. Walter, D. Dreher, M. Kok, L. Thiele, S.G. Kiama, P . Gehr, H.P . Merkle ( Zurich, Geneva, Berne, Switzerland) 149 PII: S0168-3659(01)00466-7

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Journal of Controlled Release 76 (2001) 385–387

www.elsevier.com/ locate / jconrel

Contents Volume 76 (2001)

Vol. 76, Nos. 1 –2 (11 SEPTEMBER 2001)

Research papersEffect of PSC 833 liposomes and Intralipid on the transport of epirubicin in Caco-2 cells and rat intestines

1Yu.-l. Lo, F.-i. Liu, J.-y. Cherng (Tainan, Taiwan)Protein delivery from materials formed by self-selective conjugate addition reactions

11D.L. Elbert, A.B. Pratt, M.P. Lutolf, S. Halstenberg, J.A. Hubbell (Zurich, Switzerland)Temperature-controlled content release from liposomes encapsulating Pluronic F127

27P. Chandaroy, A. Sen, S.W. Hui (Buffalo, NY, USA)Investigation of the influence of mean HPMC particle size and number of polymer particles on the release of

aspirin from swellable hydrophilic matrix tabletsP.W.S. Heng, L.W. Chan, M.G. Easterbrook, X. Li (Kent Ridge Crescent, Merchant Square, Singapore) 39

Cross-linked high amylose starch derivatives as matrices for controlled release of high drug loadings´J. Mulhbacher, P. Ispas-Szabo, V. Lenaerts, M.A. Mateescu (Montreal, Laval, Canada) 51

Evaluation of particle uptake in human blood monocyte-derived cells in vitro. Does phagocytosis activity ofdendritic cells measure up with macrophages?L. Thiele, B. Rothen-Rutishauser, S. Jilek, H. Wunderli-Allenspach, H.P. Merkle, E. Walter (Zurich,Switzerland) 59

Piroxicam delivery into human stratum corneum in vivo: iontophoresis versus passive diffusion`C. Curdy, Y.N. Kalia, A. Naik, R.H. Guy (Archamps, France, Geneve, Switzerland) 73

Toxicological evaluation of a bioadhesive nasal powder containing a starch and Carbopol 974 P on rabbit nasalmucosa and slug mucosaC. Callens, E. Adriaens, K. Dierckens, J.P. Remon (Gent, Belgium) 81

Experimental determination of the theophylline diffusion coefficient in swollen sodium-alginate membranesM. Grassi, I. Colombo, R. Lapasin (Trieste, Milan, Italy) 93

Poly(ethylene glycol)–human serum albumin–paclitaxel conjugates: preparation, characterization andpharmacokineticsF. Dosio, S. Arpicco, P. Brusa, B. Stella, L. Cattel (Turin, Italy) 107

Emulsions containing partially water-miscible solvents for the preparation of drug nanosuspensionsM. Trotta, M. Gallarate, F. Pattarino, S. Morel (Novara, Italy) 119

Dipeptide model prodrugs for the intestinal oligopeptide transporter. Affinity for and transport via hPepT1 in thehuman intestinal Caco-2 cell lineC.U. Nielsen, R. Andersen, B. Brodin, S. Frokjaer, M.E. Taub, B. Steffansen (Copenhagen, Denmark) 129

Functional feature of a novel model of blood brain barrier: studies on permeation of test compoundsA. Cestelli, C. Catania, S. D’Agostino, I. Di Liegro, L. Licata, G. Schiera, G.L. Pitarresi, G. Savettieri,V. De Caro, G. Giandalia, L.I. Giannola (Palermo, Italy) 139

Gene deliveryHydrophilic poly(DL-lactide-co-glycolide) microspheres for the delivery of DNA to human-derived macrophages

and dendritic cellsE. Walter, D. Dreher, M. Kok, L. Thiele, S.G. Kiama, P. Gehr, H.P. Merkle (Zurich, Geneva, Berne,Switzerland) 149

PII : S0168-3659( 01 )00466-7

386 Contents Volume 76 (2001)

Stability of PEI–DNA and DOTAP–DNA complexes: effect of alkaline pH, heparin and serum˜´I. Moret, J. Esteban Peris, V.M. Guillem, M. Benet, F. Revert, F. Dası, A. Crespo, S.F. Alino (Valencia,

Spain) 169A new gene delivery formulation of polyethylenimine /DNA complexes coated with PEG conjugated fusogenic

peptideH. Lee, J.H. Jeong, T.G. Park (Taejon, South Korea) 183

Calendar of Events 193

Vol. 76, No. 3 (19 OCTOBER 2001)

Research papersNon-aqueous encapsulation of excipient-stabilized spray-freeze dried BSA into poly(lactide-co-glycolide)

microspheres results in release of native protein´K.G. Carrasquillo, A.M. Stanley, J.C. Aponte-Carro, P. De Jesus, H.R. Costantino, C.J. Bosques,

K. Griebenow (San Juan, Puerto Rico, Cambridge, MA, USA) 199Poly(ethylene carbonate)s, part II: degradation mechanisms and parenteral delivery of bioactive agents

¨G.H. Stoll, F. Nimmerfall, M. Acemoglu, D. Bodmer, S. Bantle, I. Muller, A. Mahl, M. Kolopp, K. Tullberg(Basel, Switzerland) 209

Alkyl-substituted silica gel as a carrier in the controlled release of dexmedetomidineP. Kortesuo, M. Ahola, M. Kangas, T. Leino, S. Laakso, L. Vuorilehto, A. Yli-Urpo, J. Kiesvaara, M. Marvola(Turku, Helsinki, Finland) 227

Fabrication, characterization and in vitro release of paclitaxel (Taxol ) loaded poly (lactic-co-glycolic acid)microspheres prepared by spray drying technique with lipid /cholesterol emulsifiersL. Mu, S.S. Feng (Singapore, Singapore) 239

Controlled release and ocular absorption of tilisolol utilizing ophthalmic insert-incorporated lipophilic prodrugsS. Kawakami, K. Nishida, T. Mukai, K. Yamamura, J. Nakamura, T. Sakaeda, M. Nakashima, H. Sasaki(Nagasaki, Kobe, Japan) 255

Stimuli-responsive properties of conjugates of N-isopropylacrylamide-co-acrylic acid oligomers with alanine,glycine and serine mono-, di- and tri-peptidesV. Bulmus, S. Patır, S.A. Tuncel, E. Piskin (Ankara, Turkey) 265

Protein release microparticles based on the blend of poly(D,L-lactic-co-glycolic acid) and oligo-ethylene glycolgrafted poly(L-lactide)K.Y. Cho, S.H. Choi, C.-H. Kim, Y.S. Nam, T.G. Park, J.-K. Park (Daejon, Kyounggi-do, South Korea) 275

Conjugation of anti-My9 antibody to stealth monensin liposomes and the effect of conjugated liposomes on thecytotoxicity of immunotoxinM. Sudhan Shaik, N. Kanikkannan, M. Singh (Tallahassee, FL, USA) 285

Effect of protein molecular weight on release from micron-sized PLGA microspheresM. Sandor, D. Enscore, P. Weston, E. Mathiowitz (Providence, RI, Warwick, RI, USA) 297

Protein release profiles and morphology of biodegradable microcapsules containing an oily coreB.B.C. Youan, T.L. Jackson, L. Dickens, C. Hernandez, G. Owusu-Ababio (Tallahassee, FL, USA) 313

Studies on the effect of pH on the lipoidal route of penetration across stratum corneumM. Sznitowska, S. Janicki, A. Baczek (Gdansk, Poland) 327

Development and release characterization of hyaluronan–doxycycline gels based on metal coordinationT. Miyazaki, C. Yomota, S. Okada (Tokyo, Osaka, Japan) 337

Galactosylated chitosan-graft-poly(ethylene glycol) as hepatocyte-targeting DNA carrierI.K. Park, T.H. Kim, Y.H. Park, B.A. Shin, E.S. Choi, E.H. Chowdhury, T. Akaike, C.S. Cho (Suwon,Kwangju, South Korea, Yokohama, Japan) 349

1.7Absorption of water-soluble compounds with different molecular weights and [Asu ]-eel calcitonin from variousmucosal administration sitesA. Yamamoto, T. Iseki, M. Ochi-Sugiyama, N. Okada, T. Fujita, S. Muranishi (Kyoto, Japan) 369

Contents Volume 76 (2001) 387

Calendar of Events 375Author Index Volume 76 379Subject Index Volume 76 383Contents Volume 76 385