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ADVANCING EARLY DRUG DISCOVERY Icagen Corporate Headquarters 4222 Emperor Blvd, Suite 350 Durham, NC 27703 +1 919-941-5206 Email us: [email protected] Icagen-T Inc. 2090 E. Innovation Park Drive Oro Valley, AZ 85755 +1 520-544-6800 Visit us at: www.icagen.com A Target-to-Lead Partner Icagen’s integrated approach is at the core of everything we do, positioning us as a comprehensive partner across early drug discovery. Employing specific expertise in medicinal chemistry with highly-specialized methodologies in computational chemistry, ultra-high throughput screening, and drug discovery biology, we wholly support our partners to determine drug feasibility and generate viable leads with unprecedented speed. Our in-house capabilities span multiple disciplines, but are united in the common goal of advancing early drug discovery programs.

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Page 1: ADVANCING EARLY DRUG DISCOVERY (PDFs)/Icagen_IDDflyer.pdfADVANCING EARLY DRUG DISCOVERY Icagen Corporate Headquarters 4222 Emperor Blvd, Suite 350 Durham, NC 27703 +1 919-941-5206

ADVANCING EARLY DRUG DISCOVERY

Icagen Corporate Headquarters4222 Emperor Blvd, Suite 350Durham, NC 27703

+1 919-941-5206

Email us: [email protected]

Icagen-T Inc.2090 E. Innovation Park DriveOro Valley, AZ 85755

+1 520-544-6800

Visit us at: www.icagen.com

A Target-to-Lead Partner

Icagen’s integrated approach is at the core of everything we do, positioning us as a comprehensive partner across early drug discovery. Employing specific expertise in medicinal chemistry with highly-specialized methodologies in computational chemistry, ultra-high throughput screening, and drug discovery biology, we wholly support our partners to determine drug feasibility and generate viable leads with unprecedented speed. Our in-house capabilities span multiple disciplines, but are united in the common goal of advancing early drug discovery programs.

Page 2: ADVANCING EARLY DRUG DISCOVERY (PDFs)/Icagen_IDDflyer.pdfADVANCING EARLY DRUG DISCOVERY Icagen Corporate Headquarters 4222 Emperor Blvd, Suite 350 Durham, NC 27703 +1 919-941-5206

Synthetic Chemistry

Medicinal Chemistry

Selectivity Profiling

Potency/Selectivity Optimization

Computational Modeling

in vitro Pharmacology

Efficacy in Patient Cells

Animal Models

in vitro Early ADME

Human Disease Models

Mechanism of Action

Pharmacokinetics/ Pharmacodynamics

Drug Interaction/ Metabolism Studies

in silico Screening

High Throughput Screening

High Content Screening

Orthogonal Screening

Active Series Expansion

Early Discovery Lead Optimization

Target Credentialing

Patient Cell Model Development

Custom Library Creation

Assay Creation

in silico Target Assessment

Hit Identification Hit to Lead

Icagen advances early drug discovery through industry-leading experience, taking many different target classes to advanced leads.

INTEGRATED DRUG DISCOVERY