2003-2004 gihb pharmacology review 19 september 2015 3:29 am
TRANSCRIPT
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2003-2004GIHB Pharmacology
Review
April 19, 202305:33 PM
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Activated charcoal
Antidote
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Albendazole
Antihelminthic
Treatment of intestinal roundworms
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Alosetron
IBS treatment
5HT3 receptor antagonist
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Aluminum hydroxide
Antiulcer
Antacid
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Amoxicillin
Penicillin antibioticCell wall synthesis inhibitor
Antiulcer
Amino penicillinInhibits peptidoglycan cross-
linking
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Ampicillin
Penicillin antibioticCell wall synthesis inhibitor
Amino penicillinInhibits peptidoglycan cross-
linking
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Anthraquinonescascara segrada, danthron, senna
Contact cathartics
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Aprepitant dimenhydrinate
Antiemetic
Neurokinin 1 receptor antagonist
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Arsenicals
Tropical antiparasitic
Treatment of African Trypanosomiasis in CNS
Melarsoprol
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Atropine
Anticholinergic
AntimuscarinicTreatment for bradycardia,
diarrhea, cholinesterase poisoning
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Azithromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor
50S ribosome Inhibits translocation
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Balsalazide
NSAID (salicylate)
Treatment of IBD
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Bisacodyl
Contact cathartic
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Bismuth subsalicylate
AntiulcerAntidiarrheal
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Budesonide
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidInhaled OR treatment of IBD
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Calcium carbonate
Antiulcer
Antacid
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Cascara sagrada
Contact cathartic
Anthraquinone derivative
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Castor Oil
Contact cathartic
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Cimetidine
AntihistamineAntiulcer
H2 receptor antagonist
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Cisapride
Prokinetic agent
5HT4 agonist
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Clarithromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor Antiulcer
50S ribosomeInhibits translocation
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Danthron
Contact cathartic
Anthraquinone derivative
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Dexamethasone
AdrenocorticosteroidGlucocorticoidAntineoplastic
Antiemetic
Anti-inflammatory steroidNot by inhalation
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Diethylcarbamazine
Antihelminthic
Treatment of intestinaland tissue roundworms
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Dimenhydrinate
AntihistamineAntiemetic
H1 receptor antagonist
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Diphenhydramine
Classical antihistamineAntiemetic
H1 antagonist
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Diphenoxylate docusate
Antidiarrheal
Opiate
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Docusates
Lubricating laxatives
Stool softeners
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Doxycycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
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Dronabinol
Antiemetic
Cannabinoid
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Droperidol
Antiemetic
D2 receptor antagonist
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Erythromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor
50S ribosomeInhibits translocation
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Granisetron
Antiemetic
5HT3 receptor antagonist
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Infliximab
TNF inhibitor
Anti-TNF monoclonal antibody Treatment of IBD
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Iodoquinol
Antiparasitic
Treatment of protozoal infections
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Ipecac
Emetic
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Ivermectin
Antihelminthic
Treatment of intestinaland tissue roundworms
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Kaolin
Antidiarrheal
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Lactulose
Saline (osmotic) cathartic
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Lansoprazole
Antiulcer
H+/K+ ATPase inhibitor
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Loperamide
Antidiarrheal
Opiate
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Magnesium hydroxide
AntiulcerSaline (osmotic) cathartic
Antacid
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Mebendazole
Antihelminthic
Treatment of intestinal roundworms
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Meclizine
AntihistamineAntiemetic
H1 receptor antagonist
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Meglumine antimonate
Tropical antiparasitic
Organic antimonialTreatment of Leishmaniasis
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Melarsoprol
Tropical antiparasitic
Treatment of African Trypanosomiasis in CNS
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Mesalamine(5-ASA)
NSAID (salicylate)
Treatment of IBD
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Methylcellulose
Bulk laxative
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Metoclopramide
Prokinetic agentAntiemetic
D2 antagonist
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Metronidazole
AntibioticAntiparasitic
Antiulcer
AnaerobesReduction leads to intermediates
that damage DNA
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Mineral oil
Lubricating laxative
Stool softener
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Minocycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
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Misoprostol
ProstaglandinAntiulcer
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Nifurtimox
Tropical antiparasitic
Treatment of South American Trypanosomiasis; Chagas
disease
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Olsalazine
NSAID (salicylate)
Treatment of IBD
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Omeprazole/esomeprazole
Antiulcer
H+/K+ ATPase inhibitor
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Ondansetron
Antiemetic
5HT3 receptor antagonist
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Organic antimonials
Tropical antiparasitic
Treatment of Leishmaniasis
sodium stibogluconatemeglumine antimonate
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Oxytetracycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
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Pantoprazole
Antiulcer
H+/K+ ATPase inhibitor
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Paromomycin
AntiparasiticAminoglycoside antibiotic
Treatment of protozoal infections
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Pectin
Antidiarrheal
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Pentamidine
Tropical antiparasitic
Treatment of African Trypanosomiasis
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Polyethylene glycol- electolyte solution
AntidoteCathartic
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Praziquantel
Antihelminthic
Treatment of trematode (fluke) and cestode (tapeworm)
infections
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Procarbazine
Antineoplastic
MiscellaneousProbably acts as alkylating
agent
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Prochlorperazine
Antiemetic
D2 receptor antagonistPhenothiazine
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Promethazine
Classical antihistamineAntipsychotic
Antiemetic
H1 antagonist
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Pyrantel Pamoate
Antihelminthic
Treatment of intestinal roundworms
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Pyrimethamine
AntimalarialProtein and nucleic acid
synthesis inhibitor
Plasmodial dihydrofolate reductase inhibitor
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Rabeprazole
Antiulcer
H+/K+ ATPase inhibitor
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Ranitidine
AntihistamineAntiulcer
H2 receptor antagonist
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Rebamipide
Antiulcer
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Senna
Contact cathartic
Anthraquinone derivative
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Scopolamine
AnticholinergicAntiemetic
Muscarinic receptor antagonist
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Simethicone
Anti-flatulent
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Sodium bicarbonate
AntiulcerAntidote
AntacidAlkalinization of urine to treat drug toxicity (esp. barbiturates, salicylates,
methanol)
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Sodium phosphate
Saline (osmotic) cathartic
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Sodium stibogluconate
Tropical antiparasitic
Organic antimonial Treatment of Leishmaniasis
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Sucralfate
Antiulcer
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Sulfasalazine
Disease modifyinganti-rheumatic drug (DMARD)
Metabolized to sulfonamide+ salicylate (NSAID) Treatment of IBD
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Suramin
Tropical antiparasitic
Treatment of African Trypanosomiasis
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Tegaserod
IBS treatment
5HT4 receptor agonist
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Tetracycline
AntibioticBacteriostatic protein synthesis
inhibitor Antiulcer
30S ribosomePrevents aminoacyl tRNA attachment
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Thiabendazole
Antihelminthic
Treatment of intestinal roundworms